{"id":33124,"date":"2019-10-31T21:50:52","date_gmt":"2019-10-31T18:50:52","guid":{"rendered":"https:\/\/prohoster.info\/blog\/o-boevyh-inkapasitantah\/"},"modified":"2019-10-31T21:50:52","modified_gmt":"2019-10-31T18:50:52","slug":"o-boevyh-inkapasitantah","status":"publish","type":"post","link":"https:\/\/prohoster.info\/sq\/blog\/news\/o-boevyh-inkapasitantah","title":{"rendered":"P\u00ebr incapsitant\u00ebt luftarak\u00eb","gt_translate_keys":[{"key":"rendered","format":"text"}]},"content":{"rendered":"<p>P\u00ebrsh\u00ebndetje, %username%.<\/p>\n<p><noindex><a rel=\"nofollow\" href=\"https:\/\/habr.com\/ru\/users\/gjf\/\" class=\"user_link\">gjf<\/a><\/noindex> p\u00ebrs\u00ebri n\u00eb lidhje.<\/p>\n<p>Menj\u00ebher\u00eb k\u00ebrkoj falje, n\u00ebse <noindex><a rel=\"nofollow\" href=\"https:\/\/habr.com\/ru\/post\/450598\/\">artikulli i m\u00ebparsh\u00ebm<\/a><\/noindex> m\u00eb duket shum\u00eb e m\u00ebrzitshme, por n\u00eb disa \u00e7\u00ebshtje m\u00eb mungon plot\u00ebsisht ndjenja e humorit.<\/p>\n<p>Dhe k\u00ebrkoj falje, n\u00ebse kam shkat\u00ebrruar iluzionet e disa lexuesve. <\/p>\n<p>Por pas votimit do t\u00eb flasim p\u00ebr droga luftuese. Por k\u00ebto nuk jan\u00eb ndonj\u00eb preparate mitologjike q\u00eb do ta kthejn\u00eb nj\u00eb njeri t\u00eb dob\u00ebt n\u00eb nj\u00eb Ushtar Universale.<\/p>\n<p>N\u00eb t\u00eb v\u00ebrtet\u00eb nuk \u00ebsht\u00eb k\u00ebshtu.<br \/>\n<noindex><a rel=\"nofollow\" name=\"habracut\"><\/a><\/noindex><br \/>\nKur sapo fillova t\u00eb studioj tem\u00ebn, m\u00eb interesuan m\u00eb shum\u00eb inkapasitancat. Akoma: n\u00eb nj\u00ebfar\u00eb momenti njer\u00ebzimi kuptoi papritmas se n\u00ebse do t\u00eb helmonte t\u00eb gjith\u00eb me di\u00e7ka si fosgjeni dhe gazrat V \u2014 njer\u00ebzimi vet\u00eb nuk do t\u00eb mbetet! <\/p>\n<p>Inkapasitancat jan\u00eb shum\u00eb m\u00eb interesante! Sipas p\u00ebrkufizimit, \"inkapasitancat jan\u00eb substanca q\u00eb p\u00ebrkoh\u00ebsisht d\u00ebmtojn\u00eb forc\u00ebn e gjall\u00eb\". Pik\u00ebrisht \"nga q\u00ebndrimi\" \u2014 por jo p\u00ebr vdekje.<\/p>\n<p>N\u00eb jet\u00ebn time kam hasur informacione q\u00eb inkapacitancat i p\u00ebrkasin nj\u00eb numri t\u00eb madh n\u00ebngrupesh:<br \/>\n<b class=\"spoiler_title\">Nj\u00eb list\u00eb e \u00e7uditshme, q\u00eb kam gjetur n\u00eb internet<\/b><\/p>\n<ol>\n<li>Alogjen\u00ebt \u2014 substanca q\u00eb shkaktojn\u00eb dhimbje t\u00eb forta kur prekin l\u00ebkur\u00ebn. Aktualisht ka p\u00ebrb\u00ebr\u00ebs t\u00eb shitur, p\u00ebr vet\u00ebmbrojtjen e popullat\u00ebs. Shpesh kan\u00eb edhe efekt t\u00eb pik\u00ebris\u00eb. Shembuj: 1-metoksi-1,3,5-cikloheptatrien, dibenzoksazepin\u00eb, kapsaicin, morfolid i acidit pelargonik, reziniferatoksin, eter\u00ebt e forbolit, cikloheptatrien.<\/li>\n<li>Anksiogjen\u00ebt \u2014 shkaktojn\u00eb nj\u00eb sulm t\u00eb papritur paniku te njeriu. Shembuj: agonist\u00ebt e receptor\u00ebve t\u00eb holicistokinin\u00ebs tip B.<\/li>\n<li>Antikoagulant\u00ebt \u2014 ulin koagulimin e gjakut, duke shkaktuar gjakderdhje. Shembuj: supervarfarin\u00eb, p\u00ebrb\u00ebr\u00ebsit e dikumarinit.<\/li>\n<li>Attraktant\u00ebt \u2013 t\u00ebrheqin insekte ose kafsh\u00eb t\u00eb ndryshme (p.sh., t\u00eb gjakosura, t\u00eb pad\u00ebshira) te njeriu. Kjo mund t\u00eb \u00e7oj\u00eb n\u00eb nj\u00eb reaksion paniku te njeriu ose t\u00eb provokoj\u00eb sulmin e insekteve ndaj njeriut. gjithashtu mund t\u00eb p\u00ebrdoren p\u00ebr t\u00eb t\u00ebrhequr d\u00ebmtuesit n\u00eb arat e armikut. Shembull: 3,11-dimetil-2-nonakozanon (attraktanti p\u00ebr zorr\u00eb).<\/li>\n<li>Afrodiziak\u00ebt \u2014 shkaktojn\u00eb nj\u00eb rritje t\u00eb madhe t\u00eb d\u00ebshir\u00ebs seksuale. Sipas studimeve, kjo mund t\u00eb provo\u00e7onte konflikte n\u00eb nj\u00eb kolektiv ushtarak pothuajse nj\u00eb-gjinor. Shembuj: viagra, sialis.<\/li>\n<li>Noxhoret (si substanca me er\u00eb t\u00eb k\u00ebqij) \u2013 shkaktojn\u00eb largimin e njer\u00ebzve nga nj\u00eb territor ose nga nj\u00eb individ, p\u00ebrmes ndjenj\u00ebs s\u00eb neveritjes nga era e pak\u00ebndshme e vendit (ose individit). Era e pak\u00ebndshme mund t\u00eb ket\u00eb t\u00eb b\u00ebj\u00eb me substancat vet\u00eb ose produkte t\u00eb metabolizmit t\u00eb tyre. Exemple: merkaptanet, izonitrilet, selenolet, teluriti i natriumit, geosmini, benzociklopropani.<\/li>\n<li>Shkaktues t\u00eb dhimbjeve n\u00eb muskuj \u2013 shkaktojn\u00eb ndjenja t\u00eb forta dhimbjeje n\u00eb muskujt e njeriut. Exemple: aminoethet e timolit.<\/li>\n<li>Shkaktues t\u00eb humbjes s\u00eb flok\u00ebve \u2013 q\u00ebllimi i p\u00ebrdorimit \u00ebsht\u00eb t\u00eb ndikojn\u00eb n\u00eb individ\u00eb me aktivitet shoq\u00ebror, p\u00ebr t\u00eb zvog\u00ebluar t\u00ebrheqjen e jashtme. Exemple: kripra e talliumit.<\/li>\n<li>Agjent\u00eb hipotensiv\u00eb \u2014 ulin ndjesh\u00ebm presionin, duke shkaktuar kolaps ortostatik, p\u00ebr pasoj\u00eb, individi humb vet\u00ebdijen ose aft\u00ebsin\u00eb p\u00ebr t\u00eb l\u00ebvizur. Exemple: klonidin\u00eb, kanabisol, analoge t\u00eb faktor\u00ebve t\u00eb aktivizimit t\u00eb trombociteve.<\/li>\n<li>Agjent\u00eb hormonal\u00eb \u2014 ndikojn\u00eb n\u00eb shum\u00eb sisteme t\u00eb trupit n\u00eb konsentrime shum\u00eb t\u00eb vogla, gj\u00eb q\u00eb mund t\u00eb shkaktoj\u00eb ndryshime n\u00eb ndjesit\u00eb dhe gjendjen emocionale. Shpesh jan\u00eb zhvilluar forma metabolikisht stabile t\u00eb hormoneve. Exemple: insulina, hormoni adrenokortikotropik, glukokortikoid\u00ebt.<\/li>\n<li>Denaturant\u00ebt \u2014 japin shije t\u00eb pak\u00ebndshme produkteve ushqimore, rezultati i t\u00eb cilave mund t\u00eb shkaktoj\u00eb urin\u00eb n\u00eb zonat e prekura. Exemple: kripra e denatoniumit, kinin\u00eb.<\/li>\n<li>Kastrator\u00ebt \u2014 shkaktojn\u00eb kastrimin kimik (humben aft\u00ebsin\u00eb p\u00ebr riprodhim). Exemple: gossypol.<\/li>\n<li>Katatonik\u00ebt \u2014 shkaktojn\u00eb zhvillimin e katatonis\u00eb te individ\u00ebt e prekur. Zakonisht i p\u00ebrkasin nj\u00eb kategorie t\u00eb substancave psikokimike helmuese. Exemple: bulbokapnin.<\/li>\n<li>Miorelaksant\u00ebt periferik\u00eb \u2014 shkaktojn\u00eb relaksimin e plot\u00eb t\u00eb muskujve skeletor\u00eb. Mund t\u00eb shkaktojn\u00eb vdekjen p\u00ebr shkak t\u00eb relaksimit t\u00eb muskujve t\u00eb frym\u00ebmarrjes. Exemple: tubokurarin, ditilin.<\/li>\n<li>Miorelaksant\u00ebt qendror\u00eb \u2014 shkaktojn\u00eb relaksimin e muskujve skeletor\u00eb. P\u00ebr dallim nga ata periferik\u00eb, ato kan\u00eb ndikim m\u00eb t\u00eb vog\u00ebl n\u00eb frym\u00ebmarrje dhe detoxifikimi i tyre \u00ebsht\u00eb i v\u00ebshtir\u00eb. Exemple: miorelaksin, fenilglicerin, benzimidazol.<\/li>\n<li>Mokogjen\u00eb \u2014 shkaktojn\u00eb nj\u00eb p\u00ebrshpejtim t\u00eb menj\u00ebhersh\u00ebm t\u00eb zbrazjes s\u00eb fshik\u00ebz\u00ebs s\u00eb urin\u00ebs. Exemple: furosemid.<\/li>\n<li>Anestezik\u00ebt \u2013 shkaktojn\u00eb anestezi te njer\u00ebzit e sh\u00ebndosh\u00eb. N\u00eb k\u00ebt\u00eb moment, p\u00ebrdorimi i k\u00ebsaj grupi substancash \u00ebsht\u00eb i v\u00ebshtir\u00eb p\u00ebr shkak t\u00eb aktivitetit t\u00eb ul\u00ebt biologjik t\u00eb substancave t\u00eb p\u00ebrdorura. Exemple: izoflurani, halothan.<\/li>\n<li>Droga e t\u00eb v\u00ebrtet\u00ebs \u2013 shkakton te njer\u00ebzit nj\u00eb gjendje n\u00eb t\u00eb cil\u00ebn ata nuk mund t\u00eb flasin q\u00ebllimisht g\u00ebnjeshtra. Aktualisht, \u00ebsht\u00eb d\u00ebshmuar se kjo metod\u00eb nuk garanton plot\u00ebsisht sinqeritetin e individ\u00ebve dhe p\u00ebrdorimi i saj \u00ebsht\u00eb i kufizuar. Zakonisht nuk \u00ebsht\u00eb substanc\u00eb individuale, por nj\u00eb kombinim i barbiturat\u00ebve me stimulator\u00eb.<\/li>\n<li>Analgjezike narkotike \u2013 n\u00eb doza m\u00eb t\u00eb larta se ato terapeutike shkaktojn\u00eb nj\u00eb efekt immobilizues. Ato jan\u00eb n\u00eb gjendje t\u00eb shkaktojn\u00eb var\u00ebsi. Shembuj: fentanil, karfentanil, 14-metoksimetopon, etorfin, dihidroetorfin.<\/li>\n<li>Substanca q\u00eb d\u00ebmtojn\u00eb kujtes\u00ebn \u2013 shkaktojn\u00eb humbje t\u00eb p\u00ebrkohshme t\u00eb kujtes\u00ebs. Shpesh jan\u00eb toksike. Shembuj: cikloheksimid, acid doborik, shum\u00eb antikolinerik\u00eb, disa benzodiazepin\u00eb.<\/li>\n<li>Neuroleptik\u00ebt \u2013 shkaktojn\u00eb ngadal\u00ebsim motorik dhe mendor te individi. Shembuj: haloperidol, spiperon, flufhenazin.<\/li>\n<li>Inhibitor\u00eb t\u00eb pakthyesh\u00ebm t\u00eb MAO \u2013 grup substancash q\u00eb bllokojn\u00eb monoaminooksidaz\u00ebn. Si rezultat, kur konsumohen produkte me p\u00ebrmbajtje t\u00eb lart\u00eb t\u00eb aminave natyrore (djath\u00ebra, \u00e7okollat\u00eb), provokojn\u00eb nj\u00eb kriz\u00eb hipertensive. Shembuj: nialamid, pargilin.<\/li>\n<li>Shtyp\u00ebs t\u00eb vullnetit \u2013 shkaktojn\u00eb \u00e7rregullim t\u00eb aft\u00ebsis\u00eb p\u00ebr t\u00eb marr\u00eb vendime t\u00eb pavarura. Jan\u00eb substanca t\u00eb grupeve t\u00eb ndryshme. Shembuj: skopolamin.<\/li>\n<li>Prurigen\u00eb \u2013 shkaktojn\u00eb kruajtje t\u00eb padurueshme. Shembuj: 1,2-dithiocyanodethane.<\/li>\n<li>Mjetet psikotomimetike \u2013 shkaktojn\u00eb psikoza q\u00eb zgjasin p\u00ebr nj\u00ebfar\u00eb kohe, gjat\u00eb s\u00eb cil\u00ebs individi nuk \u00ebsht\u00eb n\u00eb gjendje t\u00eb marr\u00eb vendime t\u00eb p\u00ebrshtatshme. Shembuj: BZ, LSD, meskalin, DMT, DOB, DOM, kanabinoid\u00eb, PCP, psilocibin\u00eb, DET, DMGP.<\/li>\n<li>Laksativ\u00eb \u2013 shkaktojn\u00eb shpejt\u00ebsim t\u00eb papritur t\u00eb zbrazjes s\u00eb p\u00ebrmbajtjes s\u00eb zorr\u00ebve. Me veprimin e gjat\u00eb t\u00eb preparateve t\u00eb k\u00ebtij grupi, mund t\u00eb zhvillohet shterbimi i trupit. Shembuj: bisakodil.<\/li>\n<li>Substancat q\u00eb shkaktojn\u00eb lot \u2013 shkaktojn\u00eb lotim t\u00eb fort\u00eb dhe mbyllje t\u00eb qepallave, duke b\u00ebr\u00eb q\u00eb individi t\u00eb mos jet\u00eb n\u00eb gjendje t\u00eb shoh\u00eb p\u00ebrreth dhe t\u00eb humbas\u00eb aft\u00ebsin\u00eb p\u00ebr t\u00eb luftuar. Ka substanca helmuese q\u00eb p\u00ebrdoren p\u00ebr shp\u00ebrndarjen e demonstratave. Shembuj: chloracetophenone, bromacetone, bromobenzylcyanide, krip\u00ebrat e trialkyllead, ethylbromacetate, ethylidacetate, ortho-chlorobenzylidenemalononitrile (CS).<\/li>\n<li>Mjetet q\u00eb shkaktojn\u00eb gjum\u00eb \u2013 shkaktojn\u00eb flen\u00eb t\u00eb individ\u00ebve. Shembuj: flunitrazepam, barbiturat\u00eb.<\/li>\n<li>Sternit\u00ebt shkaktojn\u00eb teshtitje dhe kollitje t\u00eb pakontrolluar, duke b\u00ebr\u00eb q\u00eb personi t\u00eb heq\u00eb mask\u00ebn. Ekzistojn\u00eb agjent\u00eb t\u00eb klasifikuar. Shembuj: adamzit, difenilklorarsin, difenilcianarsin.<\/li>\n<li>Tremorgen\u00ebt shkaktojn\u00eb kontraktime spasmodike t\u00eb muskujve skeletor\u00eb. Shembuj: tremorin, oksotremorin, tremorgen\u00ebt mikotoksina.<\/li>\n<li>Fotosensibilizator\u00ebt rrisin ndjeshm\u00ebrin\u00eb e l\u00ebkur\u00ebs ndaj rrezeve ultraviolet t\u00eb diellit. Kur del n\u00eb drit\u00ebn e diellit, personi mund t\u00eb marr\u00eb djegie t\u00eb dhimbshme. Shembuj: hipericini, furokumarina.<\/li>\n<li>Emetik\u00ebt (t\u00eb vjell\u00ebs) shkaktojn\u00eb refleksin e t\u00eb vjell\u00ebs, duke b\u00ebr\u00eb q\u00eb t\u00eb jet\u00eb e pamundur t\u00eb q\u00ebndrosh me mask\u00eb. Shembuj: derivatet e apomorfin\u00ebs, enterotoksina B e stafilokokut, PHNO, derivatet e aminotetralin\u00ebs.<\/li>\n<\/ol>\n<p>Duke qen\u00eb se kjo \u00ebsht\u00eb Habr, dhe ky opus nuk e shkruan nj\u00eb doktor shkencash, gjeneral-major i ushtris\u00eb kimike, an\u00ebtar korrespodent dhe t\u00eb tjera, do ta lejoj veten t\u00eb kontestoj k\u00ebt\u00eb list\u00eb. <br \/>\n<b class=\"spoiler_title\">Mungesa do t\u00eb jet\u00eb e shkurt\u00ebr, nj\u00ebanshme, shum\u00eb jokorrekte dhe jasht\u00ebzakonisht subjektive.<\/b>\u2018Droga e s\u00eb v\u00ebrtet\u00ebs\u2019 duhet t\u00eb administrohet intravenoze \u2014 dhe gjithmon\u00eb duhet t\u00eb ket\u00eb nj\u00eb ndikim psikologjik mbi personin. Si mund t\u00eb p\u00ebrdoret kjo n\u00eb nj\u00eb situat\u00eb luftarake? Dhe \u2018shembujt\u2019 jan\u00eb shum\u00eb t\u00eb diskutuesh\u00ebm: p\u00ebr shembull \u2018kastratori\u2019 gossypol \u2014 nj\u00eb polifenol natyror, ka veti antivirale, antimykotike, anti-protozoar, antioksiduese dhe aktivitet antitumoral. Nuk kam par\u00eb askund informacion se ai p\u00ebrdoret p\u00ebr kastrimin kimik: nuk \u00ebsht\u00eb hormon si ciproteroni acetat, nga i cili madje edhe te nj\u00eb macho tipik do t\u00eb rriten gjoksat, dhe nuk \u00ebsht\u00eb neuroleptik si benperidoli, nga i cili nuk do t\u00eb d\u00ebshirosh asgj\u00eb. Duket se roli i \u2018kastrator\u00ebve\u2019 n\u00eb zvog\u00eblimin e aft\u00ebsis\u00eb luftuese ka ndryshuar shum\u00eb p\u00ebr autor\u00ebt pas historis\u00eb s\u00eb Theon Greyjoy \u2014 mir\u00eb, k\u00ebshtu \u00ebsht\u00eb, ai m\u00eb pas u tregua madje shum\u00eb i zoti.<\/p>\n<p>A do t'i trembin substancat e ndyrshme luft\u00ebtar\u00ebt? K\u00ebto i ka shkruar dikush q\u00eb nuk ka qen\u00eb kurr\u00eb n\u00eb kazerm\u00eb.<\/p>\n<p>Dhe m\u00eb shum\u00eb \u2014 skopolamina \u2014 nj\u00eb n\u00ebnshtrues i vullnetit? Buga.<\/p>\n<p>Prandaj nuk do t\u00eb p\u00ebrpiqem t\u00eb paraqes shembuj nga ky list\u00eb p\u00ebr \u00e7do grup. Ndoshta ata ekzistojn\u00eb dhe jan\u00eb t\u00eb klasifikuar, ndoshta \u2014 jan\u00eb thjesht fantazi t\u00eb autor\u00ebve q\u00eb i kan\u00eb paraqitur, ose ndoshta \u2014 thjesht nuk dua )))<\/p>\n<p>M\u00eb trishton grupi i irritant\u00ebve - kjo \u00ebsht\u00eb nj\u00eb p\u00ebrb\u00ebrje e lakrimatoreve (p\u00ebr at\u00eb q\u00eb qan) dhe sterbin\u00ebve (p\u00ebr at\u00eb q\u00eb kollitet). Nuk do t\u00eb shqyrtoj irritant\u00ebt - s\u00eb pari, ata gjithashtu kan\u00eb probleme - veprojn\u00eb p\u00ebr pak koh\u00eb, sidomos n\u00ebse e braktisin zon\u00ebn e goditjes, dhe ndonj\u00ebher\u00eb ndodhin d\u00ebshtime aksidentale, si n\u00eb CS n\u00eb Vietnam (megjithat\u00eb, pas p\u00ebrdorimit t\u00eb defoliant\u00ebve, nuk mendoj se ishte ndonj\u00eb fatkeq\u00ebsi e madhe). Megjithat\u00eb, si\u00e7 kuptova, leximet e gjata e lodhin lexuesin )<\/p>\n<p>Prandaj, %username%, le t\u00eb flasim p\u00ebr di\u00e7ka shum\u00eb m\u00eb interesante!<\/p>\n<p>N\u00eb k\u00ebt\u00eb rast nuk do t\u00eb ket\u00eb nj\u00eb hit-parad\u00eb, k\u00ebshtu q\u00eb le t\u00eb zgjedh\u00eb secili favoritin e tij.<\/p>\n<p><b class=\"spoiler_title\">Fluorotani (halotani)<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/ddc0dd2304b949a694b9d5badb3dd438.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nFluorotani \u00ebsht\u00eb m\u00eb irrituesi, m\u00eb i thjeshti dhe m\u00eb pak interesanti nga t\u00eb gjitha. Ky \u00ebsht\u00eb nj\u00eb l\u00ebng i pa ngjyrosur, i pambrojtur dhe shum\u00eb i avulluesh\u00ebm (temperatura e zierjes rreth 50\u00b0C). T\u00eb t\u00eb kujton morg.<\/p>\n<p>Fluorotani p\u00ebrdoret n\u00eb anestezi gjat\u00eb operacioneve t\u00eb ndryshme, p\u00ebrfshir\u00eb ato n\u00eb organet e barkut ose t\u00eb kraharorit, te f\u00ebmij\u00ebt dhe njer\u00ebzit e moshuar, te pacient\u00ebt me astm\u00eb bronkiale. P\u00ebrdorimi i anestezis\u00eb me fluorotan \u00ebsht\u00eb ve\u00e7an\u00ebrisht i dobish\u00ebm kur duhet t\u00eb shmanget eksitimi dhe tensionsi te paciente (p.sh., n\u00eb neurokirurgji, oftalmologji, etj.). P\u00ebr t'u futur n\u00eb anestezi, fillohet me administrimin e fluorotanit n\u00eb p\u00ebrqindje 0.5 vol. % (me oksigjen), pastaj p\u00ebr 1.5\u20133 minuta rritet deri n\u00eb 3\u20134 vol. %. P\u00ebr t\u00eb mbajtur faz\u00ebn kirurgjikale t\u00eb anestezis\u00eb, p\u00ebrdoret p\u00ebrqindja 0.5-2 vol. %.<\/p>\n<p>Gjat\u00eb p\u00ebrdorimit t\u00eb fluorotanit, nd\u00ebrgjegjja zakonisht fiket pas 1-2 minutash nga fillimi i thithjes s\u00eb avujve t\u00eb tij. Pas 3-5 minutash arrihet faza kirurgjikale e anestezis\u00eb. Pas 3-5 minutash nga ndalimi i dh\u00ebnies s\u00eb fluorotanit, pacient\u00ebt nisin t\u00eb zgjohen. Depresioni anestezike zhduket plot\u00ebsisht pas 5-10 minutash pas anestezis\u00eb s\u00eb shkurt\u00ebr dhe pas 30-40 minutash pas anestezis\u00eb s\u00eb gjat\u00eb. Eksitimi v\u00ebrehet rrall\u00eb dhe \u00ebsht\u00eb i dob\u00ebt. T\u00eb irrituara organet e frym\u00ebmarrjes nuk ndodhin fare.<\/p>\n<p>T\u00eb thuhet q\u00eb t\u00eb luash me fluorotanin nuk \u00ebsht\u00eb e men\u00e7ur, sepse n\u00eb disa raste shkakton d\u00ebmtime t\u00eb r\u00ebnda n\u00eb m\u00ebl\u00e7i (hepatiti halotan). Kryesisht hepatiti ndodh tek njer\u00ebzit mbi 40 vje\u00e7, duke u shfaqur m\u00eb shpesh te grat\u00eb se te burrat. Veprimi toksik i fluorotanit \u00ebsht\u00eb i shkaktuar jo vet\u00ebm nga ndikimi direkt, por edhe nga formimi i metabolit\u00ebve toksik\u00eb (acid tri-fluoroacetik, tri-fluoroetanol, tri-fluoroacetaldehid).<\/p>\n<p>Por, duke qen\u00eb se avujt e fluorotanit jan\u00eb rreth 6.7 her\u00eb m\u00eb t\u00eb r\u00ebnd\u00eb se ajri, ai \u00ebsht\u00eb v\u00ebn\u00eb realisht n\u00eb shqyrtim si nj\u00eb variant i \"gazit q\u00eb b\u00ebn t\u00eb flej\u00eb\", me disavantazhin se veprimi duhet t\u00eb jet\u00eb i shpejt\u00eb, sepse pas 5 minutash, kur avujt shp\u00ebrndahen, t\u00eb gjith\u00eb do t\u00eb zgjohen.<\/p>\n<p>T\u00eb nj\u00ebjtat veti ka edhe izoflurani.<br \/>\n<b class=\"spoiler_title\">Izofluran<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/dad059476f27c428b9f49c527f3e33a5.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nK\u00ebto jan\u00eb di\u00e7ka si kap\u00ebs t\u00eb nivelit fillestar. Por ato hapin Grupin e Madh dhe T\u00eb Friksh\u00ebm t\u00eb fizikant\u00ebve - substanca q\u00eb shkaktojn\u00eb \u00e7rregullime t\u00eb shkurt\u00ebr - fizike ose fiziologjike.<\/p>\n<p>Kush tjet\u00ebr kemi k\u00ebtu?<\/p>\n<p><b class=\"spoiler_title\">Apomorfin<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/955b32800982f6190a9ff800d14515fb.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nPo, apomorfin \u00ebsht\u00eb me siguri i njohur p\u00ebr ata q\u00eb kan\u00eb ndjer\u00eb ndonj\u00ebher\u00eb d\u00ebshira p\u00ebr vet\u00ebvrasje ose e kan\u00eb provuar nj\u00eb helmim t\u00eb r\u00ebnd\u00eb. Po, ky \u00ebsht\u00eb ila\u00e7i q\u00eb merret nga morfina duke vepruar mbi t\u00eb me acid klorhidrik. N\u00eb k\u00ebt\u00eb m\u00ebnyr\u00eb, hiqet lidhja oksigjenike tipike p\u00ebr alkaloid\u00ebt e morfin\u00ebs dhe si rezultat i riorganizimit molekular formohet nj\u00eb lidhje e re kat\u00ebrciklike.<\/p>\n<p>T\u00eb gjith\u00eb narkoman\u00ebt, q\u00ebndroni dhe mos vraponi n\u00eb farmaci - apomorfin, edhe pse ruan disa nga vetit\u00eb e babait t\u00eb tij, ka nj\u00eb veprim ndryshe: \u00ebsht\u00eb nj\u00eb preparat shum\u00eb i fuqish\u00ebm p\u00ebr t\u00eb vjellur. 0.01 mg\/kg shkakton ndjenjat e m\u00ebposhtme: fillimisht, ti, %username%, do t\u00eb ndihesh pak si n\u00eb det: zbardhje, djersitje t\u00eb ftoht\u00eb, nauze - n\u00ebse asnj\u00ebher\u00eb nuk ke ndier t\u00eb vjell\u00eb, at\u00ebher\u00eb p\u00ebrpara - do ta kuptosh garantuar se si \u00ebsht\u00eb. Pastaj, pas rreth 3-10 minutash, do t\u00eb fillosh t\u00eb vjell\u00ebsh menj\u00ebher\u00eb, abundsh\u00ebm dhe pa ndales\u00eb. Jo, nuk \u00ebsht\u00eb ajo \"t\u00eb vjell\u00ebsh\", si pas pirjes - jo, do t\u00eb kesh nj\u00eb mik t\u00eb bardh\u00eb, i cili gjithmon\u00eb ndodhet n\u00eb apartamentin t\u00ebnd n\u00eb nj\u00eb vend t\u00eb nderuar. Duhet ta p\u00ebrqafosh dhe ta th\u00ebrras\u00ebsh Ichthyandrin p\u00ebr rreth nj\u00eb or\u00eb - vazhdimisht, me ndonj\u00eb pushim t\u00eb rrall\u00eb. Pastaj do t\u00eb qet\u00ebsohesh - nj\u00eb dob\u00ebsi e vog\u00ebl dhe gjith\u00e7ka do t\u00eb kaloj\u00eb.<\/p>\n<p>Tani \u00ebsht\u00eb e qart\u00eb pse apomorfin p\u00ebrdoret n\u00eb tortura gjat\u00eb helmimeve?<\/p>\n<p>\u00cbsht\u00eb e qart\u00eb se ushtari i guximsh\u00ebm, i cili d\u00ebshiron t\u00eb kthehet te vendlindja, pak do t\u00eb jet\u00eb i dobish\u00ebm n\u00eb luft\u00eb. Nj\u00eb mang\u00ebsi e vetme: apomorfina duhet t\u00eb jet\u00eb e injektuar n\u00eb gjak ose e p\u00ebrtypur p\u00ebrmes hund\u00ebs. Pijet me uj\u00eb p\u00ebr efektin k\u00ebrkojn\u00eb nj\u00eb sasi t\u00eb madhe (m\u00eb shum\u00eb se 10 mg) \u2014 dhe kjo n\u00eb nj\u00eb kapsul\u00eb xhelatine me acid askorbik, p\u00ebrndryshe substanca do t\u00eb prish\u00eb n\u00eb stomak. N\u00eb luft\u00eb kjo nuk do t\u00eb jet\u00eb e mundur.<\/p>\n<p>Sidoqoft\u00eb, apomorfina shpesh p\u00ebrdoret p\u00ebr t\u00eb trajtuar alkoolist\u00ebt e zakonsh\u00ebm. Metoda e trajtimit \u00ebsht\u00eb e thjesht\u00eb: injektohet apomorfina hydrochloride n\u00ebn l\u00ebkur\u00eb n\u00eb nj\u00eb doz\u00eb nga 0,002 g deri n\u00eb 0,01 g, duke p\u00ebrshtatur individualisht doz\u00ebn q\u00eb shkakton t\u00eb vjella te ky pacient. Pas 3\u20134 minutash pas injektimit t\u00eb apomorfin\u00ebs, pacienti i jepet nj\u00eb got\u00eb me 30\u201350 ml pije alkoolike, t\u00eb cil\u00ebn ai e konsumon n\u00eb m\u00ebnyr\u00eb abuzive. N\u00eb fillim t\u00eb t\u00eb vjellave, i propozohet t\u00eb pij\u00eb nj\u00eb gll\u00ebnk\u00eb t\u00eb pijeve, pas s\u00eb cil\u00ebs ai duhet ta nuhas at\u00eb dhe ta b\u00ebj\u00eb gargara me goj\u00eb. Kur t\u00eb filloj\u00eb t\u00eb p\u00ebrkeq\u00ebsohet, dhe pacienti t\u00eb ndjej\u00eb ardhjen e t\u00eb vjellave, duhet t\u00eb pij\u00eb edhe nj\u00eb gll\u00ebnk\u00eb t\u00eb pijeve alkoolike. Zakonisht, pas 1-15 minutash nga shfaqja e t\u00eb vjellave, ndodh\u00ebn t\u00eb vjellat. Seancat kryhen 1-2 her\u00eb n\u00eb dit\u00eb. Pavlovi e duartroket.<\/p>\n<p>Ka edhe substanca t\u00eb tjera me nj\u00eb veprim t\u00eb ngjash\u00ebm. Ja nj\u00eb shembull i af\u00ebrt:<br \/>\n<b class=\"spoiler_title\">Likorini<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/ac0026afe0e73e4afa81cfacc674ad56.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nLikorini nuk merret, ai ekstrahohet: \u00ebsht\u00eb nj\u00eb alkaloid, i pranish\u00ebm n\u00eb disa bim\u00eb nga familja amaryllidaceae, ve\u00e7an\u00ebrisht n\u00eb bim\u00ebt e familjeve clivia, crinum, galanthus, ungernia.<br \/>\nKy preparat \u00ebsht\u00eb rreth 50 her\u00eb m\u00eb i dob\u00ebt se apomorfina, por shkakton t\u00eb vjella edhe n\u00eb rast t\u00eb helmimit me neuroleptik\u00eb \u2014 prandaj \u00ebsht\u00eb shum\u00eb i preferuar nga vet\u00ebvras\u00ebsit.<\/p>\n<p><b class=\"spoiler_title\">Fentanili<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/721c82e1a8690bbe520c0329b705fd95.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nKam nj\u00eb p\u00ebrkushtim personal ndaj k\u00ebsaj substance, por kjo \u00ebsht\u00eb nj\u00eb histori tjet\u00ebr. Fentanili \u00ebsht\u00eb nj\u00eb analgjezik narkotik. N\u00eb praktik\u00ebn mjek\u00ebsore p\u00ebrdoret n\u00eb form\u00ebn e citratit. Ofron nj\u00eb veprim t\u00eb fuqish\u00ebm dhe t\u00eb shpejt\u00eb analgjezik. N\u00eb rusisht \u2014 nga ai b\u00ebjn\u00eb drog\u00eb. Dhe shum\u00eb. Ashtu si nga heroina.<\/p>\n<p>P\u00ebrmes injektimit parenteral n\u00eb kafsh\u00eb, shkakton analgjezi n\u00eb doza q\u00eb p\u00ebrb\u00ebjn\u00eb mij\u00ebra-qindrat e nj\u00eb fraksioni mg\/kg. Efekti ndodh pas 2\u201310 minutash. Doza vdekjeprur\u00ebse e fentanilit p\u00ebr nj\u00eb mi n\u00eb injektim intravenoz \u00ebsht\u00eb LD50 = 3\u20135 mg\/kg. Fentanili shkakton te njeriu humbjen e ndjeshm\u00ebris\u00eb me nj\u00eb doz\u00eb orale 0,05\u20130,1 mg\/kg, ndersa me nj\u00eb doz\u00eb mbi 0,2 mg\/kg ndodhin konvulsione.<\/p>\n<p>Sigurisht, kimist\u00ebt trim kan\u00eb pushuar s\u00eb anashkalojn\u00eb fentanilin dhe po k\u00ebrkojn\u00eb aktivisht se \u00e7far\u00eb mund t\u00eb b\u00ebjn\u00eb me t\u00eb p\u00ebr ta b\u00ebr\u00eb at\u00eb m\u00eb t\u00eb shpejt\u00eb, m\u00eb t\u00eb lart\u00eb dhe m\u00eb t\u00eb fort\u00eb. Dhe duhet th\u00ebn\u00eb - arrit\u00ebn. Disa arritje m\u00eb posht\u00eb.<\/p>\n<p><b class=\"spoiler_title\">Karfentanil<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/6a8a7ee9879b1865926b5a2f4eb3d29b.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nSuksesi m\u00eb i r\u00ebnd\u00ebsish\u00ebm. \u00cbsht\u00eb nj\u00eb nga opiatet m\u00eb t\u00eb fuqishme, nj\u00eb nj\u00ebsi karfentanili \u00ebsht\u00eb 100 her\u00eb m\u00eb e fuqishme se e nj\u00ebjta sasi fentanili, 5000 her\u00eb m\u00eb e fuqishme se nj\u00eb nj\u00ebsi heroine dhe 10,000 her\u00eb m\u00eb e fuqishme se nj\u00eb nj\u00ebsi morfine. Aktiviteti analgjezike median ED50 (do t\u00eb thot\u00eb - ndikoi n\u00eb 50% t\u00eb subjekt\u00ebve) p\u00ebr k\u00ebt\u00eb substanc\u00eb kur injektohet n\u00eb vena te minjt\u00eb \u00ebsht\u00eb 0,41 mcg\/kg, doza mediane vdekjeprur\u00ebse LD50 (k\u00ebtu 50% vdiq\u00ebn) \u00ebsht\u00eb 3,39 mg\/kg, ndikimi n\u00eb trupin e njeriut fillon q\u00eb nga 1 mcg.<\/p>\n<p>Karfentanili n\u00eb koh\u00eb paqeje p\u00ebrdoret si qet\u00ebsues p\u00ebr elefant\u00eb: n\u00ebse ti, %username%, ke nj\u00eb elefant n\u00eb sht\u00ebpi, p\u00ebr ta anestezuar - e di se mjafton dy miligram karfentanili. Ky substanc\u00eb prodhohet komercialisht: preparati \u00ebsht\u00eb i pranish\u00ebm n\u00eb tregun farmaceutik me mark\u00ebn tregtare Wildnil si anestetik me veprim t\u00eb p\u00ebrgjithsh\u00ebm, i destinuar p\u00ebr kafsh\u00ebt e m\u00ebdha - aktiviteti shum\u00eb i lart\u00eb nuk parashikon p\u00ebrdorimin e saj te njer\u00ebzit. N\u00ebse je kurioz - analgjeziku m\u00eb i fuqish\u00ebm q\u00eb p\u00ebrdoret p\u00ebr q\u00ebllime mjek\u00ebsore te njer\u00ebzit aktualisht \u00ebsht\u00eb sufentanili, rreth 10-20 her\u00eb m\u00eb i dob\u00ebt se karfentanili. P\u00ebr m\u00eb tep\u00ebr, p\u00ebr kafsh\u00ebt e vogla p\u00ebrdoren edhe ohmefentanili. Dhe po, t\u00eb gjith\u00eb k\u00ebto \"shiringa fluturuese\" jan\u00eb nga kjo tem\u00eb. <\/p>\n<p>Nj\u00eb nga shembujt m\u00eb t\u00eb njohur t\u00eb p\u00ebrdorimit t\u00eb karfentanilit n\u00eb praktik\u00ebn veterinar \u00ebsht\u00eb episod i serialit dokumentar Animal Cops: Houston t\u00eb kanalit Discovery, ku u tregua se si karfentanili (i holluar n\u00eb mjalt\u00eb) u p\u00ebrdor p\u00ebr t\u00eb anestezuar nj\u00eb ari t\u00eb kafshuar p\u00ebr t\u2019u transportuar n\u00eb m\u00ebnyr\u00eb t\u00eb sigurt nga nj\u00eb pronar privat q\u00eb e keqtrajtonte at\u00eb n\u00eb Teksas Jugor n\u00eb kopshtin zoologjik t\u00eb Houston.<\/p>\n<p>Sipas disa ekspert\u00ebve, t\u00eb cilat nuk jan\u00eb konfirmuar nga strukturat ruse t\u00eb forcave t\u00eb siguris\u00eb, aerosoli me baz\u00eb karfentanil \u00ebsht\u00eb p\u00ebrdorur gjat\u00eb sulmit n\u00eb Qendren Teatrale n\u00eb Dubrovka n\u00eb Mosk\u00eb n\u00eb vitin 2002, p\u00ebr t\u00eb reduktuar mund\u00ebsin\u00eb e aktivizimit t\u00eb pajisjeve shp\u00ebrthyese nga terrorist\u00ebt. Ky p\u00ebrfundim u arrit nga fakti se sh\u00ebrbimet e urgjenc\u00ebs mjek\u00ebsore ishin udh\u00ebzuar (me vones\u00eb dhe pa zbuluar natyr\u00ebn e agjentit) t\u00eb p\u00ebrdorin antagonist\u00ebt e opioid\u00ebve. P\u00ebr shkak t\u00eb munges\u00ebs s\u00eb informacionit, mjek\u00ebt nuk mund\u00ebn t\u00eb zhvillonin nj\u00eb strategji reanimimi dhe t\u00eb siguronin nj\u00eb num\u00ebr t\u00eb mjaftuesh\u00ebm t\u00eb naloksonit dhe naltrexonit p\u00ebr ndihm\u00ebn e suksesit p\u00ebr t\u00eb gjith\u00eb t\u00eb prekurit. Duke supozuar se p\u00ebrb\u00ebr\u00ebsi i vet\u00ebm aktiv i aerosolit dremit\u00ebs ishte karfentanil, shkaku kryesor i vdekjes s\u00eb t\u00eb prekurve mund t\u00eb ket\u00eb qen\u00eb gjithashtu ndalesa e frym\u00ebmarrjes e shkaktuar nga opioid\u00ebt; n\u00eb k\u00ebt\u00eb rast, frym\u00ebmarrja artificiale e aplikuar n\u00eb vend (n\u00eb vend t\u00eb transportit n\u00eb klinika) dhe p\u00ebrdorimi i antagonist\u00ebve mund t\u00eb ken\u00eb shp\u00ebtuar jet\u00ebn e shumic\u00ebs ose t\u00eb gjith\u00eb viktimave.<\/p>\n<p>D\u00ebshiroj ta theksoj edhe nj\u00eb her\u00eb: nuk kam qen\u00eb atje, po shkruaj at\u00eb q\u00eb gjendet n\u00eb burimet e hapura, dhe prandaj do t\u00eb them se ka edhe mendime t\u00eb tjera q\u00eb:<\/p>\n<ul>\n<li>Nuk \u00ebsht\u00eb p\u00ebrdorur karfentanil, por 3-metilfentanil (do t\u00eb jet\u00eb m\u00eb posht\u00eb). <\/li>\n<li>\u00cbsht\u00eb p\u00ebrdorur fluorotane (ka qen\u00eb m\u00eb lart).<\/li>\n<li>\u00cbsht\u00eb p\u00ebrdorur BZ (do t\u00eb jet\u00eb shum\u00eb posht\u00eb).<\/li>\n<\/ul>\n<p>\nN\u00eb p\u00ebrmbledhje, %username%, n\u00ebse ke pyetje t\u00eb tjera n\u00eb k\u00ebt\u00eb drejtim \u2014 telefononi n\u00eb numrin +74952242222.<\/p>\n<p><b class=\"spoiler_title\">Alfentanil<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/1d3b45bdbecfe4ae9ec4272ffe44687c.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nAlfentanil \u00ebsht\u00eb nj\u00eb v\u00eblla shum\u00eb m\u00eb i ri i karfentanilit. N\u00eb doz\u00ebn 0,0025 mg\/kg, tek njer\u00ebzit shkaktohet tremor, dhe n\u00eb doz\u00ebn 0,175 mg\/kg ndodhi imobilizimi i njeriut pas 4\u20135 minutash pas marrjes. Raportohet se Instituti Komb\u00ebtar i Drejt\u00ebsis\u00eb n\u00eb SHBA, gjat\u00eb k\u00ebrkimit t\u00eb substancave q\u00eb mund t\u00eb imobilizojn\u00eb kriminel\u00ebt pa u shkaktuar d\u00ebm, e ka p\u00ebrdorur edhe alfentanil. Megjithat\u00eb, doli se duke e tejkaluar doz\u00ebn terapeutike me 4 her\u00eb, rreziku i ndalimit fatal t\u00eb frym\u00ebmarrjes shfaqet. N\u00eb fund, studiuesit u detyruan t\u00eb heqin dor\u00eb nga eksperimente me alfentanilin dhe t\u00eb k\u00ebrkojn\u00eb substanca m\u00eb t\u00eb sigurta. Ve\u00e7an\u00ebrisht e njohur \u00ebsht\u00eb 3-metilfentanil, i sintetizuar n\u00eb vitin 1972 \u2014 nj\u00eb narkotik dhe analgjez ekstremisht i fuqish\u00ebm, m\u00eb aktiv se heroi, nga 500\u20132000 her\u00eb. N\u00eb administrimin p\u00ebrmes inhalimit, 3-metilfentanil kalon n\u00eb nivel aktiviteti shum\u00eb psikomimetik\u00eb.<\/p>\n<p><b class=\"spoiler_title\">3-metilfentanil<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/33bae9870ca16d15c6125bcd693b0f6b.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nDuke p\u00ebrve\u00e7 karakteristikave t\u00eb derivat\u00ebve t\u00eb fentanilit, disa vendos\u00ebn t\u00eb krijojn\u00eb helm me perferans dhe prostituta \u2014 k\u00ebshtu u shfaq \u03b1-metilfentanil. Ky kimikat \u00ebsht\u00eb droga m\u00eb e keqe, m\u00eb e thjesht\u00eb p\u00ebr t'u sintetizuar midis t\u00eb gjith\u00eb derivat\u00ebve t\u00eb fentanilit. Karakteristikat: shkat\u00ebrron jet\u00ebt e atyre q\u00eb e konsumojn\u00eb dhe <noindex><a rel=\"nofollow\" href=\"https:\/\/ru.wikipedia.org\/wiki\/%D0%91%D0%B5%D0%BB%D1%8B%D0%B9_%D0%BA%D0%B8%D1%82%D0%B0%D0%B5%D1%86\">ata q\u00eb e prodhojn\u00eb.<\/a><\/noindex>. Un\u00eb principialisht nuk do t\u00eb shkruaj asgj\u00eb p\u00ebr t\u00eb. M\u00eb fal, %username%.<\/p>\n<p>Nome, p\u00ebr t\u00eb immobilizuar \u2014 nuk \u00ebsht\u00eb e nevojshme t\u00eb injektohet drog\u00eb. Nj\u00eb p\u00ebrb\u00ebr\u00ebs tjet\u00ebr q\u00eb ka veprim immobilizues \u00ebsht\u00eb:<br \/>\n<img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/9459778bcd10966f82ca600ecb86934e.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n0,001 mg\/kg shkakton dob\u00ebsi fizike, megjithat\u00eb, kalon shpejt. P\u00ebr t\u00eb dob\u00ebsuar p\u00ebrhersh\u00ebm \u2014 duhet t\u00eb konsumosh shum\u00eb: doza toksike \u00ebsht\u00eb mbi 1000 her\u00eb m\u00eb e lart\u00eb.<br \/>\nSinqerisht: kam harruar emrin e thjesht\u00eb t\u00eb zakonsh\u00ebm t\u00eb k\u00ebtij p\u00ebrb\u00ebr\u00ebsi, por e gjej formul\u00ebn. P\u00ebrdorni.<\/p>\n<p>Rritim bastet, %username%! <\/p>\n<p><b class=\"spoiler_title\">Sernil<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/2298bd6f4fbe07fd90b75430d4f4fa76.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nSernil, ose feniklidin, ose SN sipas nomenklatur\u00ebs s\u00eb sh\u00ebrbimeve nd\u00ebrkomb\u00ebtare n\u00eb doza 0,03-1 mg\/kg pas nj\u00eb periudhe t\u00eb fsheht\u00eb deri n\u00eb nj\u00eb or\u00eb fillon t\u00eb funksionoj\u00eb shum\u00eb arg\u00ebtues: ndodh nj\u00eb ndryshim periodik i gjendjes s\u00eb stimulimit dhe depresionit. Nuk di si ta p\u00ebrshkruaj k\u00ebt\u00eb gam\u00eb ndjenjash, por n\u00eb fund trupi shpejt lodhet. Ndjen nj\u00eb ndjenj\u00eb t\u00eb thell\u00eb vetmie dhe izolimi, m\u00eb pas \u2014 negativiz\u00ebm dhe armiq\u00ebsi. Pas 8-10 or\u00ebsh pas marrjes s\u00eb sernilit, simptomat nuk ndryshojn\u00eb shum\u00eb nga ato t\u00eb ngjashme me skizofrenin\u00eb.<\/p>\n<p>N\u00ebse pak e tepron, at\u00ebher\u00eb me 2 mg\/kg mund t\u00eb ndodh\u00eb katalepsia deri n\u00eb 3 dit\u00eb. Kjo \u00ebsht\u00eb kur ulet, shikon jasht\u00eb dhe nuk l\u00ebviz. Por ka dhe p\u00ebrfitime \u2014 mund t\u00eb ekspozohesh n\u00eb ndonj\u00eb galeri...<\/p>\n<p>Ky mrekulli u krijua n\u00eb vitet 1950 n\u00eb SHBA dhe madje fillimisht p\u00ebrdorej p\u00ebr q\u00ebllime mjek\u00ebsore deri n\u00eb vitin 1965. Q\u00eb nga viti 1979, p\u00ebrdorimi dhe prodhimi i sernilit \u00ebsht\u00eb ndaluar.<\/p>\n<p>P\u00ebr m\u00eb tep\u00ebr, grupi interesant i lagjes t\u00ebnde mund ta njoh\u00eb sernilin si RCP, pilul\u00ebn e paqes, pluhurin e engj\u00ebllit (Angel dust) \u2014 po, po, p\u00ebr t\u00eb k\u00ebndon \u00abAria\u00bb, HOG, Killer weed, KJ, Embalming fluid, Rocker fuel, Sherms etj.<\/p>\n<p>Sernil shum\u00eb shpejt shkakton var\u00ebsi, p\u00ebrve\u00e7 k\u00ebsaj, ky person \u00ebsht\u00eb shum\u00eb xheloz p\u00ebr burimet e tjera t\u00eb k\u00ebnaq\u00ebsive t\u00eb bot\u00ebs: n\u00eb kombinim me substanca t\u00eb tjera \u2014 p\u00ebr shembull me alkoolin, marihuan\u00ebn ose benzodiazepinat \u2014 mund t\u00eb \u00e7oj\u00eb n\u00eb kom\u00eb.<\/p>\n<p>Nj\u00eb shok dhe bashk\u00ebpun\u00ebtor i sernilit \u00ebsht\u00eb kjo:<br \/>\n<b class=\"spoiler_title\">Dikush shpresonte<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/46bcb69d54779cecdc68f98dbec7d4d3.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nKjo \u00ebsht\u00eb substanca e dyt\u00eb, p\u00ebr t\u00eb cil\u00ebn kam harruar emrin e zakoneve. Tani e di shkrimin tim t\u00eb k\u00ebqij, %username%! Besom\u00eb, kjo \u00ebsht\u00eb m\u00eb e keqe se \u00e7do helm.<\/p>\n<p>Kjo gj\u00eb n\u00eb doza 60-210 mcg\/kg vepron brenda 0.5-2 or\u00ebve n\u00ebse merret p\u00ebrmes goj\u00ebs, dhe n\u00ebse inhalohet ose injektohet \u2014 brenda 5 minutash. Mesatarisht, p\u00ebr njeriun mjafton vet\u00ebm 5 mg.<\/p>\n<p>N\u00eb rast t\u00eb prekjes simotomat jan\u00eb shum\u00eb t\u00eb ngjashme me ato t\u00eb serin\u00ebs. Shpejt pas intoksikacionit shfaqet dob\u00ebsi, marramendje, dridhje dhe ngritje muskulore, pastaj vjen nauzea, ndjesi mpirjeje n\u00eb goj\u00eb dhe \u00e7rregullim i t\u00eb folurit. Dhe tashm\u00eb pas rreth nj\u00eb ore fillon e r\u00ebnd\u00ebsishmja. Humbet mund\u00ebsia p\u00ebr t'u p\u00ebrqendruar dhe p\u00ebr t\u00eb menduar, ndjesit\u00eb e koh\u00ebs dhe hap\u00ebsir\u00ebs. Nd\u00ebrpritet koordinimi, dhe reflekset kondicionale deformohen. Dhe e r\u00ebnd\u00ebsishmja: halucinacione. Ngjyrosura. Shkencore dhe vizuale. Por fatkeq\u00ebsia \u2014 t\u00eb gjitha jan\u00eb t\u00eb frikshme. N\u00eb nj\u00eb sfond t\u00eb ndjenj\u00ebs s\u00eb vazhdueshme t\u00eb frik\u00ebs dhe tmerrit \u2014 \u00ebsht\u00eb di\u00e7ka. T\u00eb kesh frik\u00eb, t\u00eb d\u00ebgjosh dhe t\u00eb shoh\u00ebsh at\u00eb q\u00eb ke frik\u00eb, do t\u00eb ndihesh p\u00ebr 5-6 or\u00eb, dhe n\u00ebse ke fat t\u00eb kap\u00ebsh 200 mcg\/kg e m\u00eb shum\u00eb \u2014 ndodh depersonalizimi total, ti, %username%, nuk je m\u00eb %username% \u2014 por nj\u00eb krijes\u00eb e vog\u00ebl e tkurrur dhe duke trembur, q\u00eb qan, ul\u00ebrit dhe KA FRIK\u00cb. E v\u00ebrtet\u00eb, \u00e7far\u00eb arg\u00ebtimi?<\/p>\n<p>T\u00eb tilla jan\u00eb arg\u00ebtimet, sa q\u00eb substancat psikotrope m\u00eb t\u00eb njohura lidhen pik\u00ebrisht me veprimin halu\u00e7inogjenik.<\/p>\n<p>Pra, mir\u00ebseardh\u00ebt \u2014 <b class=\"spoiler_title\">LSD<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/c36ec608bc4203f2ef440b851902fedc.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nPas fjal\u00ebs \u2018LSD\u2019, p\u00ebr t'u th\u00ebn\u00eb, fshihet emri i k\u00ebtij kryevepra \u2014 N,N-dietilamidi D-acidit lisergjik. Pra, \u00ebsht\u00eb si t\u00eb t\u00eb quajn\u00eb me emrin dhe mbiemrin.<\/p>\n<p>Me t\u00eb v\u00ebrtet\u00eb, %username%, nuk e di si dhe pse m\u00eb 16 n\u00ebntor 1938, kimisti zviceran Albert Hofmann n\u00eb Bazel mori LSD-25 nga acidi lisergjik (25 \u2014 sepse ishte lidhja e 25-t\u00eb q\u00eb ai sintetizoi). Njer\u00ebzimi tashm\u00eb e dinte p\u00ebr toksicitetin e ergotoksinave nga gruri i eg\u00ebr, Arthur Stoll n\u00eb laboratorin e firm\u00ebs Sandoz kishte nxjerr\u00eb konvertimin ergotamin nga sklerociet n\u00eb vitin 1918 \u2014 por e hulumtonin at\u00eb n\u00eb drit\u00ebn e veprimit stimulues ndaj muskulatur\u00ebs s\u00eb mitr\u00ebs. Nuk mendoj se Hofmann kishte ndonj\u00eb problem me mitr\u00ebn, por sidoqoft\u00eb \u2014 LSD ai e mori. Aplaudoni at\u00eb (edhe pse ai \u00ebsht\u00eb tashm\u00eb i vdekur, por jo p\u00ebr k\u00ebt\u00eb arsye).<\/p>\n<p>Dhe, m\u00eb 19 prill 1943, Hofmann si nj\u00eb shkenc\u00ebtar i v\u00ebrtet\u00eb pranoi at\u00eb q\u00eb sintetizoi. 250 mikrogram. Rezultati: pas pak koh\u00ebsh filluan t\u00eb shfaqeshin marramendja dhe shqet\u00ebsimi. Shpejt, efekti u b\u00eb aq i fort\u00eb saq\u00eb Albert nuk mund t\u00eb formonte m\u00eb fjali koherente dhe, i v\u00ebzhguar nga asistentin e tij, i njoftuar p\u00ebr eksperimentin, u nis p\u00ebr n\u00eb sht\u00ebpi me bi\u00e7iklet\u00eb. Udh\u00ebtimi ishte interesant: ndjenjat subjetive t\u00eb Hofmannit \u2014 nj\u00eb ngasje shum\u00eb e ngadalt\u00eb \u2014 nuk p\u00ebrputheshin me objektivin: ai po ecte si nj\u00eb tibetian i stimuluar. Nd\u00ebrkoh\u00eb, bulevardi i njohur n\u00eb rrug\u00ebn p\u00ebr n\u00eb sht\u00ebpi u shnd\u00ebrrua p\u00ebr Hofmannin n\u00eb nj\u00eb piktur\u00eb t\u00eb Salvador Dalit: i dukej se nd\u00ebrtesat ishin mbuluar me nj\u00eb val\u00eb t\u00eb vog\u00ebl. <\/p>\n<p>Pas arritjes n\u00eb sht\u00ebpi, Hofmann i k\u00ebrkoi asistentit t\u00eb th\u00ebrras\u00eb mjekun dhe t\u00eb k\u00ebrkoj\u00eb qum\u00ebsht nga fqinj\u00ebt, t\u00eb cilin e kishte zgjedhur si antidot t\u00eb zakonsh\u00ebm p\u00ebr helmimet.<\/p>\n<p>Mjeku i ardhur nuk gjeti asnj\u00eb devijim te pacienti p\u00ebrve\u00e7 zgjerimit t\u00eb pupillave. Megjithat\u00eb, gjat\u00eb disa or\u00ebve, Hofmann ishte n\u00eb nj\u00eb gjendje deliriumi: i dukej se ishte i mbushur me demon\u00eb, se fqinja e tij ishte nj\u00eb shtrig\u00eb, se mobilja n\u00eb sht\u00ebpin\u00eb e tij ishte k\u00ebrc\u00ebnuese p\u00ebr t\u00eb. Pastaj ndjenja e shqet\u00ebsimit u t\u00ebrhoq, duke u z\u00ebvend\u00ebsuar nga imazhe shum\u00ebngjyr\u00ebshe n\u00eb form\u00ebn e rrethave dhe spiraleve, t\u00eb cilat nuk zhdukeshin as me syt\u00eb e mbyllur. Hofmann gjithashtu tregonte se zhurma e nj\u00eb automobili q\u00eb kalonte perceptohej nga ai si nj\u00eb imazh optik.<\/p>\n<p>M\u00eb 22 prill, ai shkroi p\u00ebr eksperimenti dhe p\u00ebrvoj\u00ebn e tij, dhe m\u00eb von\u00eb e p\u00ebrfshiu k\u00ebt\u00eb sh\u00ebnim n\u00eb librin e tij \"LSD - f\u00ebmija im i v\u00ebshtir\u00eb\".<\/p>\n<p>N\u00eb parath\u00ebnien e librit t\u00eb tij, Hofmann shkroi, nd\u00ebr t\u00eb tjera, se u b\u00eb kimist p\u00ebr shkak t\u00eb d\u00ebshir\u00ebs s\u00eb tij p\u00ebr nj\u00eb nj\u00ebsi absolute me natyr\u00ebn. Ai k\u00ebrkoi substanca q\u00eb zgjeronin aft\u00ebsit\u00eb e njeriut p\u00ebr t\u00eb perceptuar bot\u00ebn rreth tij n\u00eb gjith\u00eb plot\u00ebsin\u00eb e saj. Megjithat\u00eb, n\u00eb momentin e shkruarjes s\u00eb librit, shkenc\u00ebtari tashm\u00eb e dinte se veza e zbuluar nga ai, jo vet\u00ebm q\u00eb zgjeron vet\u00ebdijen, por gjithashtu mund t\u00eb shkat\u00ebrroj\u00eb psiken e nj\u00eb njeriu, duke \u00e7uar n\u00eb pasoja katastrofike. <\/p>\n<blockquote><p>\u00abTh\u0435 intentionally invoking of mystical experiences, particularly through LSD and similar hallucinogens, poses dangers that should not be underestimated compared to spontaneous visionary experiences. Practitioners must take into account some effects of these substances, namely their ability to influence our consciousness, the very essence of who we are. The history of LSD today sufficiently demonstrates the catastrophic consequences that can occur when the depth of its effects is underestimated and this substance is regarded as a drug that can be taken for pleasure. The improper and inappropriate use has made LSD my difficult child.\u00bb<\/p><\/blockquote>\n<p>\n<i> \u2014 \u00abLSD is my difficult child\u00bb, A. Hofmann.<\/i><\/p>\n<p>Nevertheless, since April 19, 1943, some followers refer to it as the 'Day of the Bicycle' and even celebrate it. In their own way.<br \/>\n<b class=\"spoiler_title\">Mark\u00eb n\u00eb nder t\u00eb fest\u00ebs. \u00c7far\u00eb ka n\u00eb mark\u00eb nga ana tjet\u00ebr \u2014 e gjeje?<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/bfdb01308596054dd06ecc08de5844d8.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nThe mechanism of action of LSD is quite complex. Primarily, this substance is a structural analog of serotonin, a neurotransmitter that regulates rest, sleep, and energy accumulation. The anti-serotonin action of LSD leads to hallucinations. Besides being a non-specific serotonin antagonist (a substance that blocks receptors in nerve synapses where serotonin is the mediator), LSD also has an inhibiting effect on monoamine oxidase (MAO) of serotonin, as well as MAO of other mediators \u2014 \u03b3-aminobutyric acid, histamine, and norepinephrine. In short, the effect is quite diverse and, it must be said \u2014 not fully studied.<\/p>\n<p>For some time, it was believed that studying the new substance would help understand the nature of schizophrenia, which is also characterized by serotonin-related issues. However, many scientists did not believe that psychedelic and schizophrenic psychosis were identical. Despite some common features, the hypothesis of a single nature of schizophrenia and LSD action has been disproven.<\/p>\n<p>N\u00eb nj\u00eb m\u00ebnyr\u00eb ose n\u00eb nj\u00eb tjet\u00ebr, gjat\u00eb viteve 1960, u kryen hulumtime intensive p\u00ebr LSD-n\u00eb \u2014 dhe un\u00eb po flas pik\u00ebrisht p\u00ebr studime paq\u00ebsore t\u00eb shkenc\u00ebtar\u00ebve n\u00eb universitetet e SHBA-s\u00eb dhe vendeve t\u00eb tjera. Hulumtimet m\u00eb t\u00eb njohura u zhvilluan nga Stanislav Grof dhe Timothy Leary. Ky i fundit kryesonte nj\u00eb propagand\u00eb aktive p\u00ebr k\u00ebt\u00eb substanc\u00eb psikotropike, pasi besonte se efekti i saj pozitiv tejkalonte efektet an\u00ebsore t\u00eb mundshme. P\u00ebr m\u00eb tep\u00ebr, ai iu jepte LSD disa student\u00ebve pa i njoftuar p\u00ebr emrin e saj, si\u00e7 ishte praktik\u00eb e zakonshme n\u00eb at\u00eb periudh\u00eb gjat\u00eb hulumtimit t\u00eb psikedelik\u00ebve. M\u00eb von\u00eb, Timothy Leary u ndoq aktivisht nga autoritetet, p\u00ebrfshir\u00eb p\u00ebr q\u00ebndrimin e tij agresiv p\u00ebr dobin\u00eb e \"zgjatjes s\u00eb vet\u00ebdijes\" p\u00ebr njeriun.<\/p>\n<p>N\u00eb vitin 1977, gjat\u00eb d\u00ebshmive n\u00eb senatin e SHBA-s\u00eb, drejtori i CIA-s Stansfield Turner pranoi se CIA kishte kryer nj\u00eb s\u00ebr\u00eb eksperimentesh me LSD-n\u00eb mbi njer\u00ebz pa konsensusin dhe dijenin\u00eb e tyre (programi \"MK Ultra\"). K\u00ebtyre eksperimenteve iu n\u00ebnshtruan shum\u00eb amerikan\u00eb, mes t\u00eb cil\u00ebve ishin, p\u00ebrkat\u00ebsisht, t\u00eb burgosurit, pacient\u00ebt e spitaleve psikiatrike dhe pacient\u00ebt e qendrave onkologjike, infermier\u00ebt dhe \"stafi tjet\u00ebr mjek\u00ebsor\". Disa nga subjektet e eksperimentit p\u00ebrjetuan \"simptomat e para t\u00eb shizofrenis\u00eb\".<\/p>\n<p>Nj\u00eb val\u00eb entuziazmi p\u00ebr substancat psikotropike dhe LSD-n\u00eb p\u00ebrshkoi Amerik\u00ebn, e cila kishte nj\u00eb ndikim t\u00eb madh n\u00eb formimin e kontrakultur\u00ebs s\u00eb viteve '60 dhe '70. Nj\u00eb fraz\u00eb e njohur e Dr. Leary, e cila u shnd\u00ebrrua n\u00eb moto p\u00ebr mb\u00ebshtet\u00ebsit e p\u00ebrdorimit t\u00eb psikedelik\u00ebve: \"Turn on, tune in, drop out\" (\"Aktivizo, rregullo, hiqe dor\u00eb\"). Me fjal\u00ebn \"hiqe dor\u00eb\" n\u00ebnkuptohej t\u00eb ikje nga normat konservatore dhe m\u00ebnyra e jetes\u00ebs s\u00eb shumic\u00ebs s\u00eb shoq\u00ebris\u00eb.<\/p>\n<p>N\u00eb vitin 1966, n\u00eb SHBA u ndalua prodhimi, shp\u00ebrndarja dhe p\u00ebrdorimi i LSD-s\u00eb. Substanca u ndalua p\u00ebrfundimisht madje edhe p\u00ebr hulumtime laboratorike.<br \/>\n<b class=\"spoiler_title\">Sigurisht, LSD-n\u00eb e donin njer\u00ebzit krijues.<\/b><\/p>\n<ul>\n<li>Kur The Beatles regjistruan k\u00ebng\u00ebn \"Lucy in the Sky with Diamonds\", John Lennon shpjegoi origjin\u00ebn e emrit t\u00eb k\u00ebng\u00ebs duke th\u00ebn\u00eb se kjo ishte emri i nj\u00eb vizatimi t\u00eb tij nga djali i tij Julian. Megjithat\u00eb, shum\u00eb njer\u00ebz n\u00eb k\u00ebt\u00eb em\u00ebr pan\u00eb nj\u00eb aluzion p\u00ebr drog\u00ebn LSD, pasi pik\u00ebrisht k\u00ebt\u00eb akronim e p\u00ebrb\u00ebjn\u00eb inicialet e saj, dhe BBC madje e ndaloi k\u00ebng\u00ebn p\u00ebr transmetim. M\u00eb von\u00eb, Paul McCartney tregoi se ndikimi i LSD-s\u00eb n\u00eb k\u00ebt\u00eb k\u00ebng\u00eb ishte mjaft i qart\u00eb.<\/li>\n<li>P\u00ebrkrah\u00ebs t\u00eb LSD-s\u00eb ishin shkenc\u00ebtar\u00eb t\u00eb njohur si Francis Crick \u2014 nj\u00eb nga njoh\u00ebsit e struktur\u00ebs dhe funksioneve t\u00eb ADN-s\u00eb dhe Stanislav Grof, i cili u angazhua me psikologjin\u00eb transpersonale. Po ashtu, ila\u00e7in e p\u00ebrdor\u00ebn Steve Jobs dhe Bill Gates. Jobs e p\u00ebrshkruan eksperienc\u00ebn e tij me LSD si \"nj\u00eb nga dy ose tre gj\u00ebrat m\u00eb t\u00eb r\u00ebnd\u00ebsishme q\u00eb kam b\u00ebr\u00eb n\u00eb jet\u00eb\". P\u00ebrve\u00e7 k\u00ebsaj, Jobs vdiq nga kanceri i pankreasit, nd\u00ebrsa Gates \u00ebsht\u00eb nj\u00eb nga rekordmen\u00ebt p\u00ebr shum\u00ebn e parave t\u00eb dhuruara p\u00ebr bamir\u00ebsi. Me siguri kjo nuk ka lidhje.<\/li>\n<li>\u00cbsht\u00eb nj\u00eb fakt i njohur se LSD-ja u p\u00ebrdor \"p\u00ebr frym\u00ebzim\" nga shkrimtar\u00eb t\u00eb njohur bot\u00ebror\u00eb si Aldous Huxley (\"Nj\u00eb bot\u00eb e re e mrekullueshme\"), Kurt Vonnegut (\"Krevat i mac\u00ebs\"), Ken Kesey (\"Fluturoj mbi gjethe e kukulle\"), si dhe muzikant\u00eb si John Lennon, Syd Barrett, Jim Morrison e t\u00eb tjer\u00eb.<\/li>\n<li>Po ashtu, n\u00eb filmin \"Pasqyra e zez\u00eb. Brandashmyg\", heroja me shokun e tij p\u00ebrjetojn\u00eb efektin e LSD-s\u00eb q\u00eb ishte shum\u00eb e ngjashme me t\u00eb v\u00ebrtet\u00ebn.<\/li>\n<\/ul>\n<p>Por le t\u00eb kthehemi te tema jon\u00eb. N\u00eb momentin e zbulimit t\u00eb LSD-s\u00eb, p\u00ebr ushtar\u00ebt dhe sh\u00ebrbimet speciale kishte nj\u00eb list\u00eb t\u00eb gjer\u00eb t\u00eb substancave t\u00eb ndryshme me efekte t\u00eb ngjashme: meskalin\u00eb, psilocibin\u00eb, TMA, THC, nalorfin, garmin, DOM, DMT, acid ibotenik\u2026 Edhe N,N-dimetilamidi i acidit acetik \u2014 dhe ai, n\u00eb 400 mg\/kg, shkakton depresion, humbje orientimi, halu\u00e7inacione vizuale, delirium dhe letargji \u2014 p\u00ebr m\u00eb tep\u00ebr, me siguri, p\u00ebr 7 dit\u00eb!<\/p>\n<p>Por, \u00e7do mendim ndaloi te LSD. Pse?<\/p>\n<ul>\n<li>P\u00ebr nj\u00eb fluturim t\u00eb besuesh\u00ebm mjafton 0,1-0,2 mg p\u00ebr nj\u00eb person t\u00eb qet\u00eb dhe 0,3-0,5 mg p\u00ebr nj\u00eb t\u00eb dehur (po, sapo ashtu!). KJO \u00cbSHT\u00cb SHUM\u00cb PAK! Prandaj, n\u00eb vendet interesante nuk shiten pilula LSD \u2014 shiten marka, q\u00eb duke i l\u00ebpir\u00eb garanton marrjen e doz\u00ebs s\u00eb nevojshme.<\/li>\n<li>LSD mir\u00eb zgjidhet n\u00eb uj\u00eb (n\u00eb form\u00ebn e tartaratit) dhe \u00ebsht\u00eb mjaft e q\u00ebndrueshme.<\/li>\n<li>Doza vdekjeprur\u00ebse \u00ebsht\u00eb rreth 100 mg p\u00ebr person, q\u00eb \u00ebsht\u00eb 500-1000 her\u00eb m\u00eb e lart\u00eb se sa doza efektive. \u00cbsht\u00eb e v\u00ebshtir\u00eb t\u00eb vdes\u00ebsh (nd\u00ebrsa, p\u00ebr N,N-dimetilamid t\u00eb acidit acetik, p\u00ebr t\u00eb cilin p\u00ebrmenda m\u00eb her\u00ebt, zgjohet 1 nga 3 personave).<\/li>\n<li>Nuk ka efekt kumulativ.<\/li>\n<li>Nuk ka var\u00ebsi - t\u00eb pakt\u00ebn fiziologjike.<\/li>\n<li>\u00bbKalon\u00ab minimum pes\u00eb or\u00eb \u2014 maksimum dy dit\u00eb.<\/li>\n<\/ul>\n<p>\nPra, ila\u00e7i jo vet\u00ebm q\u00eb hyri n\u00eb histori, por u miratua edhe si nj\u00eb arm\u00eb me nj\u00eb kod t\u00eb qart\u00eb dhe t\u00eb kuptuesh\u00ebm LSD. Po ashtu, u sintetizuan analoge! Megjithat\u00eb, t\u00eb gjitha d\u00ebshtuan.<br \/>\n<b class=\"spoiler_title\">Alternatives to LSD (in parentheses their hallucinogenic activity relative to LSD in %)<\/b><\/p>\n<ul>\n<li>2-bromo-LSD (7%, the effect appears only in 2% of subjects, 1.5 times more active as an anti-serotonin agent than LSD, abbreviation \u2014 BOL);<\/li>\n<li>lysergic acid amide (0%);<\/li>\n<li>dimethylamide of lysergic acid (10%);<\/li>\n<li>monoethylamide of lysergic acid (5-10%);<\/li>\n<li>morpholide of lysergic acid (30%);<\/li>\n<li>1-acetyl-LSD (100%, but the duration of action is 2-3 times shorter, and the vegetative effects are more pronounced, designation \u2014 ALD-52);<\/li>\n<li>1-methyl-LSD (36%, 4 times more active than LSD in terms of anti-serotonin activity);<\/li>\n<li>1-methoxy-LSD (66%);<\/li>\n<li>pyrrolidide of lysergic acid (5%).<\/li>\n<\/ul>\n<p>The drawback of LSD was apparent: its synthesis required ergot, which had to be cultivated, and it provided little lysergic acid \u2014 the product was expensive. A search began for something that would be at least as good. And they found it!<br \/>\n<b class=\"spoiler_title\">BZ<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/b903a71fb69a7eaba9e909d3695d164b.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nNo, %username%, 'BZ' has no relation to any sounds of organic origin. And the fact that 'BZ' appears as '\u0418\u042f' due to a layout error is just a coincidence. Probably.<\/p>\n<p>BZ \u2014 3-hinuklidyl ether of benzoic acid \u2014 is a psychotomimetic from the group of glycolates. <br \/>\nIt was invented by the Swiss pharmaceutical company Hoffman-LaRoche in 1951 \u2014 the company was researching antispasmodics for treating gastrointestinal diseases. And what turned out to be unsuitable for ulcers turned out to be very suitable for other purposes (just like with Viagra, by the way). <\/p>\n<p>During this time, the United States military was searching for potential non-lethal psychoactive substances that incapacitate, including psychedelic drugs like LSD and THC, dissociative drugs like ketamine and phencyclidine, powerful opioids like fentanyl, and several glycolate anticholinergic agents. And luck favored them. <\/p>\n<p>Initially, the substance was designated as 'TK', but when it was standardized by the army in 1961, it received the NATO code name 'BZ'. The agent became commonly known as 'Buzz' due to this abbreviation and the effects it had on the mental state of volunteer subjects in scientific studies at Edgewood Arsenal in Maryland.<\/p>\n<p>N\u00eb vitin 1962, n\u00eb baz\u00ebn ushtarake Pine Bluff (Arkansas), u aktivizua nj\u00eb instalacion p\u00ebr prodhimin e substanc\u00ebs BZ n\u00eb shkall\u00eb industriale. Efikasiteti i saj luftarak u vler\u00ebsua gjat\u00eb testeve n\u00eb terren, q\u00eb p\u00ebrfunduan n\u00eb vitin 1966. <\/p>\n<p>Duke qen\u00eb se BZ \u00ebsht\u00eb kristale t\u00eb bardha me pik\u00eb shkrirjeje 190 \u00b0C, me avullim t\u00eb ul\u00ebt dhe stabilitet t\u00eb lart\u00eb termik, u p\u00ebrdor\u00ebn bomba kaset\u00eb q\u00eb shp\u00ebrndanin fishek\u00eb piroteknik\u00eb \"me avuj\" me BZ n\u00eb nj\u00eb sip\u00ebrfaqe prej rreth 1.2 hektar\u00ebsh. Po ashtu, ishin n\u00eb dispozicion \"gjenerator\u00eb\" t\u00eb mbushur me 5-6 kg BZ. Mund\u00ebsi t\u00eb tjera p\u00ebr infektimin me fragmente, plumba dhe t\u00eb tjera ishin gjithashtu t\u00eb shqyrtuara.<\/p>\n<p>BZ vepron si aerosol n\u00eb koncentrime rreth 110 mg*min\/l \u2014 dhe \u00ebsht\u00eb n\u00eb t\u00eb v\u00ebrtet\u00eb e v\u00ebshtir\u00eb t\u00eb vras\u00ebsh me k\u00ebt\u00eb substanc\u00eb, \u00ebsht\u00eb v\u00ebrejtur se grupi i rrezikut p\u00ebrfshin t\u00eb moshuarit, f\u00ebmij\u00ebt dhe njer\u00ebzit me s\u00ebmundje t\u00eb rrug\u00ebve t\u00eb frym\u00ebmarrjes.<\/p>\n<p>Fillimi \u00ebsht\u00eb i zakonsh\u00ebm: zgjerimi i pupilave, that\u00ebsi n\u00eb goj\u00eb, rritje e rrahjeve t\u00eb zemr\u00ebs. Pas 30-60 minutash ndodh akti kryesor i dram\u00ebs: dob\u00ebsimi i v\u00ebmendjes dhe kujtes\u00ebs, r\u00ebnia e reagimeve ndaj stimulimeve t\u00eb jashtme, nj\u00eb deprimim i shprehur dhe \u00e7rregullim i orientimit n\u00eb ambientin p\u00ebrreth. Pas 1-4 or\u00ebsh v\u00ebrehen takikardi t\u00eb forta, konfuzion dhe humbje kontakti me bot\u00ebn p\u00ebrreth. Halucinacionet jan\u00eb aq t\u00eb forta saq\u00eb i pafat nuk mund t\u00eb kuptoj\u00eb se \u00e7far\u00eb po ndodh n\u00eb t\u00eb v\u00ebrtet\u00eb dhe \u00e7far\u00eb \u00ebsht\u00eb thjesht imagjinat\u00eb. Kjo \u00ebsht\u00eb shum\u00eb funny, %username%. Nuk do ta besosh, v\u00ebrtet.<\/p>\n<p>N\u00eb fund zhvillohet nj\u00eb negativiz\u00ebm agresiv: njeriu b\u00ebn t\u00eb kund\u00ebrt\u00ebn e asaj q\u00eb i ofrohet. \u00c7udit\u00ebrisht, shum\u00eb shpesh - me shp\u00ebrthime zem\u00ebrimi. Kjo \u00e7menduri zgjat deri n\u00eb 4-5 dit\u00eb, nd\u00ebrsa \u00e7rregullimet mbet\u00ebse - deri n\u00eb 2-3 jav\u00eb. Mund t\u00eb ndodhi humbje e pjesshme ose e plot\u00eb e kujtes\u00ebs. <\/p>\n<p>Mekanizmi i veprimit t\u00eb BZ \u00ebsht\u00eb po aq kompleks sa ai i LSD-s\u00eb. BZ \u00ebsht\u00eb antagonist i receptor\u00ebve muskarin\u00eb t\u00eb acetikolin, pra n\u00eb thelb ai \u00ebsht\u00eb nj\u00eb kolinolitik, q\u00eb pengon transmetimin e impulsave nervore q\u00eb p\u00ebrfshijn\u00eb acetikolin \u2014 po, po, %username%, pik\u00ebrisht si VX, por ka nuanca. Nuanca \u00ebsht\u00eb raparti i lart\u00eb i doz\u00ebs toksike ndaj asaj aktive: p\u00ebr BZ ky raport \u00ebsht\u00eb rreth 40 her\u00eb (nga 32 deri n\u00eb 384 her\u00eb), pra n\u00eb thelb veprimi i BZ \u00ebsht\u00eb nj\u00eb helmim shum\u00eb-vet\u00ebm pak. N\u00eb p\u00ebrmbledhje, atje vet\u00eb djali e thyen k\u00ebmb\u00ebn, por dizajni, dimidrol dhe taren (aprofen) jan\u00eb v\u00ebllez\u00ebr sipas mekanizmit t\u00eb veprimit me BZ. Ndoshta nuk jan\u00eb t\u00eb af\u00ebrt, por sigurisht jan\u00eb kush\u00ebrinj.<\/p>\n<p>Ka nj\u00eb p\u00ebrmendje t\u00eb nj\u00eb rasti t\u00eb p\u00ebrdorimit t\u00eb substanc\u00ebs gjat\u00eb luft\u00ebs n\u00eb Vietnam, por p\u00ebr rezultatet raportohet vet\u00ebm se ato \"ishin t\u00eb k\u00ebnaqshme.\"<\/p>\n<p>Mendohet se Paul Robeson \u00ebsht\u00eb helmuar me BZ n\u00eb vitin 1961, gj\u00eb q\u00eb shkaktoi nj\u00eb episod halucinacionesh dhe depresioni t\u00eb thell\u00eb.<\/p>\n<p>N\u00eb shkurt t\u00eb vitit 1998, ministria e mbrojtjes e Britanis\u00eb s\u00eb Madhe akuzoi Irakun p\u00ebr ruajtjen e nj\u00eb sasie t\u00eb madhe t\u00eb agjentit antikolinergjik \"Agjenti 15\". Agjenti 15 supozohej t\u00eb ishte kimikisht ose i identik me BZ, ose ngusht\u00eb i lidhur me t\u00eb, dhe ruhej n\u00eb sasi t\u00eb m\u00ebdha deri dhe gjat\u00eb Luft\u00ebs n\u00eb Gjirin Persik. Megjithat\u00eb, pas luft\u00ebs CIA arriti n\u00eb p\u00ebrfundimin se Iraku nuk kishte akumuluar ose nuk kishte arm\u00ebzuar agjentin 15.<\/p>\n<p>N\u00eb janar 2013, nj\u00eb p\u00ebrfaq\u00ebsues i paidentifikuar i administrat\u00ebs amerikane, duke iu referuar nj\u00eb telegrami t\u00eb panjohur t\u00eb Departamentit t\u00eb Shtetit amerikan, deklaroi se \"kontaktet siriane tregojn\u00eb bindsh\u00ebm se agjenti 15, nj\u00eb kimikat halucinogjen i ngjash\u00ebm me BZ, ishte p\u00ebrdorur n\u00eb Homs.\" Megjithat\u00eb, n\u00eb p\u00ebrgjigje t\u00eb k\u00ebtyre raporteve, nj\u00eb p\u00ebrfaq\u00ebsues zyrtar i K\u00ebshillit t\u00eb Siguris\u00eb Komb\u00ebtare t\u00eb SHBA-s\u00eb tha: \"Raportet q\u00eb kemi par\u00eb nga mediat p\u00ebr incidentet e supozuara me arm\u00eb kimike n\u00eb Siri nuk p\u00ebrputhen me at\u00eb q\u00eb ne e konsiderojm\u00eb t\u00eb v\u00ebrtet\u00eb n\u00eb lidhje me programin sirian t\u00eb arm\u00ebve kimike.\" Substanca kimike gjithashtu supozohej t\u00eb ishte p\u00ebrdorur n\u00eb sulmet n\u00eb Ghouta n\u00eb gusht 2013.<\/p>\n<p>M\u00eb 14 prill 2018, ministri i jasht\u00ebm i RF-s\u00eb, Sergei Lavrov, njoftoi se ekspert\u00ebt nga qendra zvicerane e analizes radiologjike dhe kimike n\u00eb qytetin Shpice, t\u00eb cil\u00ebt analizuan mostrat nga Organizata p\u00ebr Ndales\u00ebn e Arm\u00ebve Kimike n\u00eb vendin e helmin t\u00eb Sergeit dhe Yulias Skripal n\u00eb Salisbury, gjet\u00ebn n\u00eb k\u00ebto mostra gjurm\u00eb t\u00eb BZ. M\u00eb 18 prill, n\u00eb nj\u00eb mbledhje t\u00eb k\u00ebshillit t\u00eb ekzekutiv t\u00eb OZA, drejtori i p\u00ebrgjithsh\u00ebm i saj, Ahmet \u00dcz\u00fcmc\u00fc, shpjegoi se prekursorja e BZ ishte p\u00ebrdorur si nj\u00eb most\u00ebr kontrolli p\u00ebr t\u00eb verifikur cil\u00ebsin\u00eb e pun\u00ebs s\u00eb laborator\u00ebve dhe nuk kishte lidhje me mostrat nga Salisbury.<\/p>\n<p>Si\u00e7 raportohet, nga 1988-1990 t\u00eb gjitha rezervat e BZ n\u00eb SHBA u shkat\u00ebrruan s\u00eb bashku me prodhimin industrial. Tani, prodhimi eksperimental i vet\u00ebm n\u00eb planet, i vendosur n\u00eb qytetin Edgewood (SHBA), lejon prodhimin e deri n\u00eb 20 ton\/n\u00eb vit, ndon\u00ebse jasht\u00eb SHBA-s\u00eb, kapacitetet totale prodhuese nuk arrijn\u00eb as 1 ton\/n\u00eb vit, pasi problema e marrjes efikase t\u00eb prekursorit t\u00eb tij \u2014 3-hinuklidol \u2014 nuk \u00ebsht\u00eb zgjidhur gjat\u00eb gjith\u00eb k\u00ebsaj kohe. K\u00ebshtu flitet, nuk e di. Por e di se ka pasur p\u00ebrpjekje p\u00ebr z\u00ebvend\u00ebsim \u2014 m\u00eb e njohura \u00ebsht\u00eb Ditrani.<br \/>\n<b class=\"spoiler_title\">Ditrani \u2014 n\u00eb t\u00eb v\u00ebrtet\u00eb nj\u00eb p\u00ebrzierje me k\u00ebt\u00eb p\u00ebrb\u00ebrje<\/b><img decoding=\"async\" alt=\"P\u00ebr incapsitant\u00ebt luftarak\u00eb\" src=\"\/wp-content\/uploads\/2019\/05\/53981fa5911bc29d262169b3a8040308.jpg\" style=\"display:block;margin: 0 auto;\" \/><br \/>\n<br \/>\nKonsiderohet se n\u00eb nj\u00eb doz\u00eb prej 5-15 mg, kjo p\u00ebrzierje shkakton simptoma t\u00eb ngjashme me BZ, q\u00eb zhvillohen brenda nj\u00eb ore.<\/p>\n<p>Aktualisht, nuk ka medikamente psikotrope q\u00eb jan\u00eb n\u00eb armatimin e vendeve t\u00eb bot\u00ebs. Por duke v\u00ebzhguar disa ngjarje masive n\u00eb vendet fqinje dhe jo aq fqinje \u2014 dyshoj shum\u00eb se \u00ebsht\u00eb k\u00ebshtu. Ndoshta nuk ndodhen n\u00eb duar t\u00eb ushtrive, por sh\u00ebrbimet e fshehta sigurisht q\u00eb punojn\u00eb.<\/p>\n<p>Pra, kjo \u00ebsht\u00eb historia q\u00eb rezultoi. <\/p>\n<p>Do ta shohim n\u00ebse do t\u2019i p\u00eblqej\u00eb, %username%. K\u00ebt\u00eb her\u00eb nuk do t\u00eb ket\u00eb votim \u2014 e gjitha do t\u00eb tregoj\u00eb renditja e artikullit.<\/p>\n<p>Fatkeq\u00ebsisht, t\u00eb shtun\u00ebn do t\u00eb filloj\u00eb nj\u00eb tjet\u00ebr periudh\u00eb udh\u00ebtimesh t\u00eb gjata dhe jo aq t\u00eb gjata \u2014 dhe p\u00ebr k\u00ebt\u00eb arsye koha p\u00ebr krijimtari do t\u00eb jet\u00eb e vog\u00ebl \u2014 do t\u00eb hyj n\u00eb nj\u00eb pushim krijues tjet\u00ebr. Dhe meqen\u00ebse koha \u00ebsht\u00eb e shkurt\u00ebr, por tani n\u00eb mendje kam vet\u00ebm nj\u00eb tregim m\u00eb shum\u00eb ose m\u00eb pak t\u00eb formuar p\u00ebr fosforin e verdh\u00eb dhe aksidentin pran\u00eb Lvivit q\u00eb lidhet me t\u00eb, n\u00ebse doli q\u00eb un\u00eb ende jam i interesant \u2014 do ta ndaj k\u00ebt\u00eb histori me ty.<\/p>\n<p>Por n\u00ebse jo \u2014 \u00e7far\u00eb do t\u00eb thot\u00eb, u mundova.<\/p>\n<p>Suksese dhe mos u s\u00ebmuresh! As fizikisht, as psikikisht\u2026<br \/>\n<br \/>Burimi: <a content=\"nofollow\" rel=\"nofollow\" href=\"https:\/\/habr.com\/ru\/post\/450756\/\">habr.com<\/a><\/p>","protected":false,"gt_translate_keys":[{"key":"rendered","format":"html"}]},"excerpt":{"rendered":"<p>\u041f\u0440\u0438\u0432\u0435\u0442, %username%. gjf \u043e\u043f\u044f\u0442\u044c \u043d\u0430 \u0441\u0432\u044f\u0437\u0438. \u0421\u0440\u0430\u0437\u0443 \u043f\u0440\u043e\u0448\u0443 \u043f\u0440\u043e\u0449\u0435\u043d\u0438\u044f, \u0435\u0441\u043b\u0438 \u043f\u0440\u0435\u0434\u044b\u0434\u0443\u0449\u0430\u044f \u0441\u0442\u0430\u0442\u044c\u044f \u043f\u043e\u043a\u0430\u0437\u0430\u043b\u0430\u0441\u044c \u0442\u0435\u0431\u0435 \u0441\u043b\u0438\u0448\u043a\u043e\u043c \u0441\u043a\u0443\u0447\u043d\u043e\u0439, \u043d\u043e \u0432 \u043d\u0435\u043a\u043e\u0442\u043e\u0440\u044b\u0445 \u0432\u043e\u043f\u0440\u043e\u0441\u0430\u0445 \u0443 \u043c\u0435\u043d\u044f \u043d\u0430\u043f\u0440\u043e\u0447\u044c \u043f\u0440\u043e\u043f\u0430\u0434\u0430\u0435\u0442 \u0447\u0443\u0432\u0441\u0442\u0432\u043e \u044e\u043c\u043e\u0440\u0430. \u0418 \u043f\u0440\u043e\u0448\u0443 \u043f\u0440\u043e\u0449\u0435\u043d\u0438\u044f, \u0435\u0441\u043b\u0438 \u0440\u0430\u0437\u0440\u0443\u0448\u0438\u043b \u0438\u043b\u043b\u044e\u0437\u0438\u0438 \u043d\u0435\u043a\u043e\u0442\u043e\u0440\u044b\u0445 \u0447\u0438\u0442\u0430\u0442\u0435\u043b\u0435\u0439. \u041d\u043e \u043f\u043e \u0438\u0442\u043e\u0433\u0430\u043c \u0433\u043e\u043b\u043e\u0441\u043e\u0432\u0430\u043d\u0438\u044f \u043c\u044b \u043f\u043e\u0433\u043e\u0432\u043e\u0440\u0438\u043c \u043e \u0431\u043e\u0435\u0432\u043e\u0439 \u043d\u0430\u0440\u043a\u043e\u0442\u0435. \u041d\u043e \u044d\u0442\u043e \u043d\u0435 \u043a\u0430\u043a\u0438\u0435-\u0442\u043e \u043c\u0438\u0444\u0438\u0447\u0435\u0441\u043a\u0438\u0435 \u043f\u0440\u0435\u043f\u0430\u0440\u0430\u0442\u044b, \u043a\u043e\u0442\u043e\u0440\u044b\u0435 \u0441\u0434\u0435\u043b\u0430\u044e\u0442 \u0438\u0437 \u0445\u0438\u043b\u043e\u0433\u043e \u0431\u043e\u0442\u0430\u043d\u0430 \u0423\u043d\u0438\u0432\u0435\u0440\u0441\u0430\u043b\u044c\u043d\u043e\u0433\u043e [&hellip;]<\/p>\n","protected":false,"gt_translate_keys":[{"key":"rendered","format":"html"}]},"author":1,"featured_media":24870,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[702],"tags":[],"class_list":["post-33124","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-news"],"aioseo_notices":[],"aioseo_head":"\n\t\t<!-- All in One SEO 5.0.2 - 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